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Understanding Oxadiazolothiazinone Biological Properties: Negative Inotropic...
We present a series of oxadiazolothiazinones, selective inotropic agents on isolated cardiac tissues, devoid of chronotropy and vasorelaxant activity. Functional and binding data for the precursor of...
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Tianagliflozin, IND filed by Tianjin Institute of Pharmaceutical research
Tianagliflozin, taigeliejing, 6-deoxydapagliflozin Molecular Formula: C21H25ClO5 Molecular Weight: 392.8732 g/mol IND Filing…Tianjin Institute of Pharmaceutical research Tianjin Institute Of...
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BMS 986120
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PF 06650808
. PF 06650808 $PFE compound inspired by auristatins ALL DATA COMING……… /////////PF 06650808
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GLPG 1690
GLPG 1690 2-[[2-ethyl-6-[4-[2-(3-hydroxyazetidin-1-yl)-2-oxoethyl]piperazin-1-yl]-8-methylimidazo[1,2-a]pyridin-3-yl]-methylamino]-4-(4-fluorophenyl)-1,3-thiazole-5-carbonitrile $GLPG compound for...
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PF 06650833
. Picture credit….Bethany Halford PF 06650833 MFC18H20FN3O4, MW361.37 1-{[(2S,3S,4S)-3-ethyl-4-fluoro-5-oxopyrrolidin-2-yl]methoxy}-7-methoxyisoquinoline-6-carboxamide 6-Isoquinolinecarboxamide,...
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LY 2922470
LY 2922470 as per WO2013025424A1 LY 2922470 Picture credit….Bethany Halford (3S)-3-[4-[[5-[(8-methoxy-3,4-dihydro-2H-quinolin-1-yl)methyl]thiophen-2-yl]methoxy]phenyl]hex-4-ynoic acid...
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Tripeptide Glycyl-L-Prolyl-L-Glutamate (Gly-Pro-Glu or GPE)
Gly-Pro-Glu Synonym: GPE, Glycyl-prolyl-glutamic acid, (1-3)IGF-1 Pfizer (Originator) Neuren Pharmaceuticals (Originator) Glypromate; glycine-proline-glutamate (neuroprotectant), Neuren CAS Number...
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Synthesis of pyrrolidinone derivatives from aniline, an aldehyde and diethyl...
Green Chem., 2016, Advance Article DOI: 10.1039/C6GC00157B, Paper Hamideh Ahankar, Ali Ramazani, Katarzyna Slepokura, Tadeusz Lis, Sang Woo Joo In this study, we reported a simple and efficient route...
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New patent, Lomitapide mesylate , Zydus Cadila Healthcare Ltd, US 20160083345,
Lomitapide mesylate Was developed and launched by Aegerion, under license from the University of Pennsylvania (which acquired rights from BMS). US-20160083345 Sanjay Jagdish DESAI Brij KHERA Jagdish...
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New patent, WO 2016042573, Acitretin, Emcure Pharmaceuticals Ltd
Acitretin PDT PATENT US4105681 WO-2016042573 Process for preparation of acitretin Emcure Pharmaceuticals Ltd EMCURE PHARMACEUTICALS LIMITED [IN/IN]; an Indian company at EMCURE HOUSE, T-184, MIDC.,...
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WO 2016042441, Mankind Research Centre, Silodosin, New patent
WO 2016042441, Mankind Research Centre, Silodosin, New patent WO-2016042441 Mankind Research Centre MANKIND RESEARCH CENTRE [IN/IN]; 191-E, Sector 4-II, IMT-Manesar, Haryana 122050 (IN) A novel...
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EDQM adopts revised monograph for WFI allowing non-destillation techniques
In a press release the EDQM has announced that the new monograph draft on Water for Injection (169) had been adopted. Read on to learn more about the production of WFI with membrane systems....
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QP Education and Qualification – What is needed?
We are frequently asked about the educational requirements in order to become a Qualified Person in Europe. Comprehensive educational modules are offered, especially in the UK. These training courses...
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DS-1040, Activated thrombin activatable fibrinolysis (TAFIa) inhibitor
DS-1040 Daiichi Sankyo Co Ltd Ischemic stroke (2S)-5-amino-2-[[1-(4-methylcyclohexyl)imidazol-4-yl]methyl]pentanoic acid 1H-Imidazole-4-propanoic acid,...
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AUNP-12 from Aurigene Discovery Technologies Limited
AUNP-12 AUR-012; Aurigene-012; NP-12, Aurigene; PD-1 inhibitor peptide (cancer), Aurigene; PD-1 inhibitor peptide (cancer), Aurigene/ Pierre Fabre; W-014A Company Aurigene Discovery Technologies...
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CRD 1152, CURADEV PHARMA PRIVATE LTD
Several candidates……One is …..CRD1152 ONE OF THEM IS CRD 1152 Kynurenine pathway regulators (solid tumors) Compound 2 CAS1638121-21-7 US159738837 N3-(3-Chloro-4- fluorophenyl) furo[2,3- c]pyridine-2,3-...
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GDC-0919; NLG-919; RG-6078
MF C18H22N2O MW: 282.17321 GDC-0919; NLG-919; RG-6078, GDC0919; GDC-0919; GDC 0919; NLG919; NLG 919; NLG-919; RG6078; RG-6078; RG 6078. 1-cyclohexyl-2-(5H-imidazo[5,1-a]isoindol-5-yl)ethanol CAS...
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CFG 920, Novartis Scientists team up with Researchers at Aurigene, Bangalore,...
CFG920, Inhibitor Of Prostate Cancer With Fewer Cardiac Side Effects Cas 1260006-20-9 Novartis Target: CYP17/CYP11B2 Disease: Castration-resistant prostate cancer MF C14H13ClN4O MW: 288.0778 Elemental...
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